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Amphetamine is thought to inhibit monoamine oxidase, whereas the flexibility of amphetamine and its metabolites to inhibit numerous P450 isozymes and various enzymes has not been adequately elucidated. In vitro experiments with human microsomes indicate insignificant inhibition of CYP2D6 by amphetamine and minimal inhibition of CYP1A2, 2D6, and 3A4